Hurevich, M. ; Swed, A. ; Joubran, S. ; Cohen, S. ; Freeman, N. S. ; Britan-Rosich, E. ; Briant-Longuet, L. ; Bardy, M. ; Devaux, C. ; Kotler, M. ; et al. Rational Conversion Of Noncontinuous Active Region In Proteins Into A Small Orally Bioavailable Macrocyclic Drug-Like Molecule: The Hiv-1 Cd4:Gp120 Paradigm. BIOORGANIC & MEDICINAL CHEMISTRY 2010, 18, 5754-5761.